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SB 218078, Tocris Bioscience™
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Quantity:
1 mg
10 mg
Description
Inhibitor of checkpoint kinase 1 (Chk1) that displays selectivity over other protein kinases (IC50 values are 15, 250 and 1000 nM for Chk1, cdc2 and PKC respectively). Abrogates G2 cell cycle arrest caused by γ-irradiation and topoisomerase I inhibition. Potentiates cytotoxicity of DNA-damaging drugs, enhancing the efficacy of some chemotherapeutics.
Specifications
Specifications
Quantity | 1 mg |
Formula Weight | 393.39 |
Percent Purity | >98% |
Chemical Name or Material | SB 218078 |
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