CAS RN 803712-79-0
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Tocris Bioscience™ Obatoclax Mesylate
Inhibitor of Bcl-2 family members (IC50 values are 1.11 - 7 μM); antiapoptotic
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Obatoclax Mesylate, MedChemExpress
MedChemExpress Obatoclax Mesylate (GX15-070 Mesylate), a BH3 mimetic, is a pan-BCL-2 family proteins inhibitor with a Ki of 220 nM for BCL-2. Obatoclax Mesylate induces autophagy-dependent cell death and targets cyclin D1 for proteasomal degradation. Obatoclax Mesylate has anti-cancer and broad-spectrum antiparasitic activity.